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    江苏宇田医药有限公司

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    Intermediate

    Contrast agent series

    Product name

    CAS Number

     5-Amino-2,4,6-Triodoisophthalolyl Chloride 37441-29-5
     5-Amino-N-(2,3-dihydroxypropyl)-2,4,6-triiodoisophthalamide Acid 111453-32-8
     5-(Acetamido)-N,N'-bis(2,3-dihydroxypropyl)-2,4,6-triiono-1,3-benzenedicarboxamide 31127-80-7
     N,N'-Bis(2,3-dihydroxypropyl)-5-[(hydroxyacetyl)amino]-2,4,6-triiodo-1,3-benzenedicarboxamide 77868-40-7
      5-Amino-N,N'-bis(2,3-dihydroxypropyl)-2,4,6-triiodo-1,3-benzenedicarboxamide 76801-93-9
     5-Amino-N,N'-bis(2,3-dihydroxypropyl)isophthalamide 203515-86-0
     N,N'-Bis(2,3-dihydroxypropyl)-5-nitro-1,3-benzenedicarboxamide 76820-34-3

    Atorvastatin Calcium Intermediate

    Product name

    CAS Number

     (4R-cis)-1,1-dimethylethyl-6-[2-[2-(4-fluorophenyl)-3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrol-1-yl]ethyl]-2,2-dimethyl-1,3-dioxane-4-acetate 125971-95-1
     (4R,cis)-1,1-dimethylethyl-6-aminoethyl-2,2-dimethyl-1,3-dioxane-4-acetate 125995-13-3
     (4R-cis)-1,1-Dimethylethyl-6-Cyanomethyl-2,2-dimethyl-1,3-dioxane-4-acetate 125971-94-0

    Rosuvastatin calcium Intermediate

    Product name

    CAS Number

     6-[(1E)-2-[4-(4-Fluorophenyl)-6-(1-methylethyl)-2-[methyl(methylsulfonyl)amino]-5-pyrimidinyl]ethenyl]-2,2-dimethyl-1,3-dioxane-4-acetic acid 1,1-dimethylethyl ester 289042-12-2
     [4-(4-Fluorophenyl)-6-isopropyl-2-(N-methylmethylsulfonamido)-pyrimidin-5-yl)methyl]triphenylpho 885477-83-8
     N-[5-(Diphenyl-phosphinoylmethyl)-4-(4-fluoro-phenyl)-6-isopropyl-pyrimidin-2-yl]-N-methyl-methanesulfonamide 289042-10-0
     4-(4-Fluorophenyl)-6-isopropyl-2- [(N-methyl-N- methylsulfony)amino]pyrimidine-5-yl-methanol 147118-36-3
     4R-Cis)-6-Hydroxymethyl-2,2-dimethyl-1,3-dioxane-4-acetic acid 1,1-dimethylethyl est 124655-09-0
     (4R-cis)-6-[(acetyloxy)methyl]-2,2-dimethyl-1,3-dioxane-4-acetic acid, t-butyl ester 154026-95-6

    Ivabradine Hydrochloride Intermediate

    Product name

    CAS Number

     (3,4-Dimethoxyphenyl)acetic acid 93-40-3
     7,8-Dimethoxy-1,3-dihydro-2H-3-benzazepin-2-one 73942-87-7
     7,8-Dimethoxy-3-(3-iodopropyl)-1,3-dihydro-2H-3-benzazepin-2-one 148870-57-9
     7,8-DiMethoxy-3-(3-chloropropyl)-1,3-dihydro-2H-3-benzazepin-2-one 85175-59-3
     4,5-Dimethoxy-1-cyanobenzocyclobutane 35202-54-1
     (1S)-4,5-Dimethoxy-1[(methylamino)methyl]benzocyclobutane hydrochloride 866783-13-3

    Silodosin Intermediate

    Product name

    CAS Number

     2-(2-(2,2,2-trifluoroethoxy)phenoxy)ethyl Methanesulfonate 160969-03-9
     5-[(2R)-2-aminopropyl]-1-[3-(benzoyloxy)propyl]-2,3-dihydro-7-carbonitrile -1H-indole (2R,3R)-2,3-dihydroxybutanedioate 239463-85-5

    MPT

    Product name

    CAS Number

     6,7-dihydro-6-mercapto-5H-Pyrazolo[1,2-a][1,2,4]triazolium chloride 153851-71-9

    Side chain for meropenem

    Product name

    CAS Number

     (2S,4S) -2-(dimethylaminocarbonyl)-4-mercapto-1- (p-nitrobenzyloxycarbonyl)-1-pyrrolidine 96034-64-9

    ASPC

    Product name

    CAS Number

     4-Nitrobenzyl (2S,4S)-4-acetylthio-2-[[N-sulfamoyl-N-(tert-butoxycarbonyl)amino]methyl]pyrrolidine-1-carboxylate 491878-06-9

    Parecoxib sodium Intermediate

    Product name

    CAS Number

      N-[4-(5-methyl-3-phenyl-oxazol-4-yl)phenyl]sulfonylpropanamide; 198470-84-7
      4-(5-METHYL-3-PHENYL-4-ISOXAZOLYL)BENZENESULFONAMIDE 181695-72-7
      5-Methyl-3,4-diphenyl 37928-17-9
     1,2-diphenyl-ethanon 451-40-1

    Sacubitril series Intermediate

    Product name

    CAS Number

     (alphaR,gammaS)-gamma-[(3-Carboxy-1-oxopropyl)amino]-alpha-methyl-[1,1'-biphenyl]-4-pentanoic acid 4-ethyl ester calcium salt 1369773-39-6
     (2R,4S)-ethyl 5-([1,1'-biphenyl]-4-yl)-4-amino-2-methylpentanoate hydrochloride 149690-12-0
     (2R,4S)-5-([1,1'-biphenyl]-4-yl)-4-((tert-butoxycarbonyl)amino)-2-methylpentanoic acid 1012341-50-2
     (R)-tert-butyl (1-([1,1'-biphenyl]-4-yl)-3-hydroxypropan-2-yl)carbamate 1426129-50-1
     4-Bromobiphenyl 92-66-0

    1,4-butanedisulfonate

    Product name

    CAS Number

     Butane-1,4-disulfonic acid 27665-39-0

    1-(2-Aminophenyl)-ethanone

    Product name

    CAS Number

     1-(2-aminophenyl)ethanone 551-93-9

    Abiraterone acetate series

    Product name

    CAS Number

     17-Iodoandrosta-5,16-dien-3beta-acetate ester 114611-53-9
     diethyl(3-pyridyl)borane 89878-14-8

    Empagliflozin Intermediate

    Product name

    CAS Number

     (3S)-3-[4-[(2-Chloro-5-iodophenyl)methyl]phenoxy]tetrahydro-furan 915095-94-2
     (3S)-3-[4-[(5-Bromo-2-chlorophenyl)methyl]phenoxy]tetrahydro-furan 915095-89-5
     S-3-hydroxytetrahydrofuran 86087-23-2

    Aprepitant Intermediate

    Product name

    CAS Number

     3-Chloromethyl-1,2,4-triazolin-5-one 252742-72-6
     (2R,3S)-2-{(1R)-1-[3,5-Bis(trifluoromethyl)phenyl]ethoxy}-3-(4-fluorophenyl)morpholine hydrochloride 171482-05-6
      (R)-1-[3,5-Bis(trifluoromethyl)phenyl]ethanol 127852-28-2
     4-Benzyl-2-hydroxy-morpholin-3-one 287930-73-8
     (R)-4-Benzyl-2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)morpholin-3-one 287930-75-0
     1M 4-fluorophenylmagnesium bromide 352-13-6

    Linezolid Intermediate

    Product name

    CAS Number

     3-Fluoro-4-morpholin-4-ylphenyl)carbamic acid benzyl ester 168828-81-7
     S)-N-[2-(Acetyloxy)-3-chloropropyl]acetamide 183905-31-9

    Acalatinib Intermediate

    Product name

    CAS Number

     4-[8-amino-3-(2S)-2-pyrrolidinylimidazo[1,5-a]pyrazin-1-yl]-N-2-pyridinyl-Benzamide 1420478-90-5
     N-Pyridin-2-yl-4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-benzamide 1383385-64-5
     [4-[(Pyridin-2-yl)carbamoyl]phenyl]boronic acid 850568-25-1
     (2S)-2-(8-amino-1-bromoimidazo[1,5-a]pyrazin-3-yl)-1-Pyrrolidinecarboxylic acid phenylmethyl ester 1420478-88-1
     (3-Chloropyrazin-2-yl)Methanamine hydrochloride 939412-86-9

    Entecavir Intermediate

    Product name

    CAS Number

      Dess-Martin periodinane 87413-09-0
     6-Benzylguanine 19916-73-5
     2-Amino-1,9-dihydro-9-[(1S,3R,4S)-4-(benzyloxy)-3-(benzyloxymethyl)-2-methylenecyclopentyl]-6H-purin-6-one 142217-81-0
     (1S,2S,3S,5S)-3-(benzyloxy)-5-(6-(benzyloxy)-2-(tritylamino)-9H-purin-9-yl)-2-((benzyloxy)methyl)cyclopentanol 1345339-53-8
     (1S,2S,3S,5S)-3-(benzyloxy)-5-(6-(benzyloxy)-2-(((4-methoxyphenyl)diphenylmethyl)amino)-9H-purin-9-yl)-2-((benzyloxy)methyl)cyclopentanol 142217-78-5
     (1S,2S,3S,5S)-5-(2-Amino-6-(benzyloxy)-9H-purin-9-yl)-3-(benzyloxy)-2-(benzyloxymethyl)cyclopentanol 142217-77-4
     (1S-trans)-2-[(Phenylmethoxy)methyl]-3-cyclopenten-1-ol 110567-21-0

    Roxadustat Intermediate

    Product name

    CAS Number

     4-Hydroxy-1-methyl-7-phenoxy-3-isoquinolinecarboxylic acid methyl ester 1421312-34-6
     Methyl 4-hydroxy-7-phenoxyisoquinoline-3-carboxylate 1455091-10-7
     5-phenoxyisobenzofuran-1(3H)-one 57830-14-5

    Febuxostat series Intermediate

    Product name

    CAS Number

     Ethyl 2-(3-cyano-4-isobutoxyphenyl)-4-methyl-5-thiazolecarboxylate 160844-75-7
     Ethyl 2-(3-cyano-4-hydroxyphenyl)-4-methylthiazole-5-carboxylate 161798-02-3
     Ethyl 2-(3-formyl-4-hydroxyphenyl)-4-methylthiazole-5-carboxylate 161798-01-2

    Lesinurad

    Product name

    CAS Number

      3H-1,2,4-Triazole-3-thione, 5-amino-4-(4-cyclopropyl-1-naphthalenyl)-2,4-dihydro- 878671-96-6
     Acetic acid, 2-((4-(4-cyclopropyl-1-naphthalenyl)-4H-1,2,4-triazol-3-yl)thio)-, methyl ester 1533519-85-5
      4-(4-cyclopropylnaphthalen-1-yl)-1H-1,2,4-triazole-5(4H)-thione 1533519-84-4
      Naphthalene, 1-cyclopropyl-4-isothiocyanato- 878671-95-5
     4-cyclopropylnaphthalen-1-aMine hydrochloride 1533519-92-4

    Sofosbuvir Intermediate

    Product name

    CAS Number

     Cytidine, N-benzoyl-2'-deoxy-2'-fluoro-2'-Methyl-, 3',5'-dibenzoate, (2'R) 817204-32-3
     (2'R)-2'-Deoxy-2'-fluoro-2'-methyluridine 863329-66-2
     (2R,3R,4R)-3- (benzoyoxy)-4-fluoro-4-methyl-5-oxotetrahydrofuran-2yl)methyl Benzoate 874638-80-9

    Abemaciclib Intermediate

    Product name

    CAS Number

     6-(2-chloro-5-fluoro-4-pyriMidinyl)-4-fluoro-2-Methyl-1-(1-Methylethyl)- 1H-BenziMidazole 1231930-42-9
     5-((4-Ethylpiperazin-1-yl)methyl)pyridin-2-amine 1180132-17-5
     6-Bromo-4-fluoro-1-isopropyl-2-methyl-1H-benzo[d]imidazole 1231930-33-8

    Ribociclib Intermediate

    Product name

    CAS Number

     2-chloro-7-cyclopentyl-N,N-dimethyl-7H-pyrrolo[2,3-d]pyrimidine-6-carboxamide 1211443-61-6
     2-chloro-7-cyclopentyl-7H-pyrrolo[2,3-d]pyrimidine-6-carboxylic acid 1211443-58-1

    Moxifloxacin Hydrochloride Intermediate

    Product name

    CAS Number

     (S,S)-2,8-Diazabicyclo[4.3.0]nonane 151213-40-0
     1-Cyclopropyl-6,7-difluoro-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid ethyl ester 112811-71-9
     1-cyclopropyl-6,7-difluoro-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid 112811-72-0

    Irinotecan Intermediate

    Product name

    CAS Number

     1-Chlorocarbonyl-4-piperidinopiperidine hydrochloride 143254-82-4
     7-Ethyl-10-hydroxycamptothecin 86639-52-3

    4-Chlorophenoxyacetyl chloride

    Product name

    CAS Number

     4-Chlorophenoxyacetyl chloride 4122-68-3


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